(E)-XS-060, CAS 2787626-06-4

(E)-XS-060, CAS 2787626-06-4
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MEXHY-149085A-0
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MedChemExpress

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Product Description: (E)-XS-060 is an isomer of XS-060. XS-060 is a RXRα antagonist. XS-060 inhibits pRXRα-PLK1 interaction. XS-060 induces RXRα-dependent mitotic arrest. XS-060 exhibits good antitumor activity against breast cancer, lung adenocarcinoma, and liver cancer[1].

Formula: C20H18N2O3

References: [1]Chen J, et al. Discovery of bipyridine amide derivatives targeting pRXRα-PLK1 interaction for anticancer therapy. Eur J Med Chem. 2023 Jun 5;254:115341.

CAS Number: 2787626-06-4

Molecular Weight: 334.37

Research Area: Cancer

Target: RAR/RXR
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Artikelnummer MEXHY-149085A-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-149085A-0
Verpackungseinheit Get quote
Mengeneinheit STK
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