AX-15836, CAS 2035509-96-5

Shelf life (days): 1460

Info: An ERK5 inhibitor (IC50 = 8 nM); selective for ERK5 over a panel of 100 other kinases at 1 µM; inhibits ERK5 autophosphorylation in HeLa cells at 1 µM; induces apoptosis in combination with ivermectin in A375 spheroids at 1 µM; decreases skin thickness and scaling in a mouse model of imiquimod-induced allergic skin inflammation at 15 mg/kg per day

Formulation: A solid

Formal Name: 2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-11-(methylsulfonyl)-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one

Purity: ≥98%

Formula Markup: C32H40N8O5S

Formula Weight: 648.77692

CAS Number: 2035509-96-5

• Artikelnummer: CAY28774-5
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 28774-5
• Verpackungseinheit: 5 mg
• Mengeneinheit: STK