Shelf life (days): 730
Info: A cell-permeable, ATP-competitive inhibitor of VprBP that blocks phosphorylation of histone 2A at Thr120 in DU-145 human prostate cancer cells (IC50 = 500 nM); strongly suppresses the proliferation of DU-145 cells, which overexpress VprBP, both in vitro and in xenograft tumors in mice
Formulation: A crystalline solid
Formal Name: 2-(5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl)hydrazone 1H-indole-3-carboxaldehyde
Purity: ≥95%
Formula Markup: C19H17N5S
Formula Weight: 347.4
CAS Number: 294193-86-5