GR 113808 (Standard), CAS 144625-51-4

Product Description: GR 113808 (Standard) is the analytical standard of GR 113808. This product is intended for research and analytical applications. GR 113808 is a potent and highly selective 5-HT4 receptor antagonist (pKb= 8.8). GR 113808 shows 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors[1].

Formula: C19H27N3O4S

References: [1]Gale JD, et al. GR113808: a novel, selective antagonist with high affinity at the 5-HT4 receptor.Br J Pharmacol. 1994 Jan;111(1):332-8./[2]Spohn SN, et al.Protective Actions of Epithelial 5-Hydroxytryptamine 4 Receptors in Normal and Inflamed Colon.Gastroenterology. 2016 Nov;151(5):933-944.e3.

CAS Number: 144625-51-4

Molecular Weight: 393.50

Research Area: Inflammation/Immunology; Neurological Disease

Target: 5-HT Receptor;Reference Standards

• Artikelnummer: MEXHY-103152R-0
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-103152R-0
• Verpackungseinheit: Get quote
• Mengeneinheit: STK