Product Description: 3-IN-PP1 is a protein kinase D (PKD) inhibitor. 3-IN-PP1 has potent pan-PKD inhibitory activity for PKD1, PKD2 and PKD3 with IC50 values of 108, 94 and 108 nM, respectively. 3-IN-PP1 also is a broad spectrum anticancer agent and has inhibition of several tumor cells growth. 3-IN-PP1 can be used for the research of cancer[1].
Applications: Cancer-Kinase/protease
Formula: C17H18N6
References: [1]Philippe Gilles, et al. Design, synthesis and biological evaluation of pyrazolo[3,4-d]pyrimidine-based protein kinase D inhibitors. Eur J Med Chem
CAS Number: 2227110-54-3
Molecular Weight: 306.37
Compound Purity: 99.58
Research Area: Cancer
Solubility: DMSO : 100 mg/mL (ultrasonic)
Target: PKD