Product Description: AZD3458 is a potent and remarkably selective PI3Kγ inhibitor with pIC50s of 9.1, 5.1, PI3Kγ, PI3Kα, PI3Kβ, and PI3Kδ, respectively[1].
Applications: Metabolism-sugar/lipid metabolism
Formula: C20H23N3O4S2
References: [1]Pemberton N, et al. Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3-Kinase (PI3K)-γ Inhibitors. J Med Chem. 2018 Jun 28;61(12):5435-5441.
CAS Number: 2132961-46-5
Molecular Weight: 433.54
Compound Purity: 99.71
Research Area: Cancer; Metabolic Disease; Inflammation/Immunology
Solubility: DMSO : 250 mg/mL (ultrasonic)
Target: PI3K