BAY-6035, CAS 2247890-13-5

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: (2S)-1-(3-azabicyclo[3.1.0]hex-3-ylcarbonyl)-N-(2-cyclopropylethyl)-2,3,4,5-tetrahydro-2-methyl-4-oxo-1H-1,5-benzodiazepine-7-carboxamide

Purity: ≥95%

Formula Markup: C22H28N4O3

Formula Weight: 396.48288

CAS Number: 2247890-13-5

Notes: BAY-6035 is an inhibitor of SET and MYND domain-containing protein 3 (SMYD3). It is 100-fold selective for SMYD3 over other histone methyltransferases. BAY-6035 inhibits methylation of MEKK2 peptide in a cell-free assay and in cells (IC50s = 88 and 70 nM, respectively). See the Structural Genomic Consortium (SGC) website for more information.

• Artikelnummer: CAY25925-5
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 25925-5
• Verpackungseinheit: 5 mg
• Mengeneinheit: STK