BAY-876, CAS 1799753-84-6

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: N4-[1-[(4-cyanophenyl)methyl]-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]-7-fluoro-2,4-quinolinedicarboxamide

Purity: ≥98%

Formula Markup: C24H16F4N6O2

Formula Weight: 496.4

CAS Number: 1799753-84-6

Notes: BAY-876 is a potent and selective inhibitor of glucose transporter 1 (Glut1) with IC50 values of 2, 10,800, 1,670, and 290 nM for Glut1, Glut2, Glut3, and Glut4, respectively, in CHO cells expressing human recombinant receptors.{38214} It shows low metabolic clearance and has high permeability in vitro. In vivo, BAY-876 displays low plasma clearance and high oral bioavailability in rats and dogs.

• Artikelnummer: CAY19961-10
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 19961-10
• Verpackungseinheit: 10 mg
• Mengeneinheit: STK