BAY-899, CAS 2471967-92-5

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: N-[2-(4-fluorophenoxy)-5-pyrimidinyl]-5-(4-fluorophenyl)-7,8-dihydro-1,6-naphthyridine-6(5H)-carboxamide

Purity: ≥98%

Formula Markup: C25H19F2N5O2

Formula Weight: 459.5

CAS Number: 2471967-92-5

Notes: BAY-899 is an antagonist of the luteinizing hormone receptor (LHR; IC50s = 185 and 46 nM for the human and rat receptors, respectively).{51892} It is selective for LHR over thyroid-stimulating hormone (TSH) and follicle-stimulating hormone (FSH) receptors (IC50s = 24 and >16 µM, respectively, for the human receptors) and a panel of 25 G protein-coupled receptors (GPCRs) at 10 µM. BAY-899 (12.5 mg/kg per day) reduces serum levels of estradiol in female rats.

• Artikelnummer: CAY41716-25
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 41716-25
• Verpackungseinheit: 25 mg
• Mengeneinheit: STK