CCF642, CAS 346640-08-2

CCF642, CAS 346640-08-2
Artikelnummer
MEXHY-100430-10.1
Verpackungseinheit
10 mM/1 ml
Hersteller
MedChemExpress

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Product Description: CCF642 is a potent protein disulfide isomerases (PDI) inhibitor with an IC50 of 2.9 μM. CCF642 causes acute endoplasmic reticulum (ER) stress in multiple myeloma cells accompanied by apoptosis-inducing calcium release. CCF642 has broad anti-multiple myeloma activity[1].

Applications: Cancer-Kinase/protease

Formula: C15H10N2O4S3

References: [1]Vatolin S et al. Novel Protein Disulfide Isomerase Inhibitor with Anticancer Activity in Multiple Myeloma. Cancer Res. 2016 Jun 1;76(11):3340-50.

CAS Number: 346640-08-2

Molecular Weight: 378.45

Compound Purity: 98.0

Research Area: Cancer

Solubility: DMSO : ≥ 30 mg/mL

Target: Apoptosis;PDI
Mehr Informationen
Artikelnummer MEXHY-100430-10.1
Hersteller MedChemExpress
Hersteller Artikelnummer HY-100430-10.1
Verpackungseinheit 10 mM/1 ml
Mengeneinheit STK
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