Shelf life (days): 1460.0
Formulation: A solid
Formal Name: N1-[(S)-(3-chloro-2-pyridinyl)(2,2-difluoro-1,3-benzodioxol-4-yl)methyl]-N2-[4-methoxy-6-(1-piperazinyl)-1,3,5-triazin-2-yl]-4-(methylsulfonyl)-1,2-benzenediamine
Purity: ≥98%
Formula Markup: C28H27ClF2N8O5S
Formula Weight: 661.080406
CAS Number: 2565705-02-2
Notes: DOT1L-IN-4 is an inhibitor of the non-SET domain-containing methyltransferase DOT1L (IC50 = 0.11 nM).{65149} It is selective for DOT1L over a panel of 11 additional histone methyltransferases at 5 µM.