DREADD Agonist 21, CAS 56296-18-5

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: 11-(1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine

Purity: ≥98%

Formula Markup: C17H18N4

Formula Weight: 278.4

CAS Number: 56296-18-5

Notes: DREADD agonist 21 activates hM3Dq (EC50 = 1.7 nM), a designer receptor exclusively activated by designer drugs (DREADD) derived from the human muscarinic acetylcholine M3 receptor.{30413} It does not agonize the hM3 receptor and displays relatively weaker binding affinities for serotonin 5-HT2A, 5-HT2C, α1A-adrenergic, and histamine H1 receptors (Kis = 66, 170, 280, and 6 nM, respectively).{30413}

• Artikelnummer: CAY18907-1
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 18907-1
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK