Ezatiostat, CAS 168682-53-9

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: (2R)-L-?-glutamyl-S-(phenylmethyl)-L-cysteinyl-2-phenyl-glycine, 1,3-diethyl ester

Purity: ≥98%

Formula Markup: C27H35N3O6S

Formula Weight: 529.7

CAS Number: 168682-53-9

Notes: Ezatiostat is an inhibitor of glutathione S-transferase pi 1-1 (GSTP1-1; Ki = 0.4 µM).{27891} It is selective for GSTP1-1 over GSTα and GSTµ family GSTs (Kis = 20-75 µM). Ezatiostat also inhibits the protein-protein interaction between GSTP1-1 and JNK1. In vivo, ezatiostat (75 mg/kg) increases the number of circulating white blood cells in Gstp1 wild-type, but not Gstp1-/-, mice.

• Artikelnummer: CAY16248-5
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 16248-5
• Verpackungseinheit: 5 mg
• Mengeneinheit: STK