BET-IN-12, CAS 1800343-11-6

BET-IN-12, CAS 1800343-11-6
Artikelnummer
MEXHY-150516S-1
Verpackungseinheit
1 mg
Hersteller
MedChemExpress

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Product Description: BET-IN-12 is an orally avtive inhibitor of bromodomain and extra-terminal (BET) with an IC50 of 0.9 nM for BRD4[1].

Applications: Cancer-programmed cell death

Formula: C30H29D3FN5O2

References: [1]Hill, Matthew D., et al. Development of BET Inhibitors as Potential Treatments for Cancer: Optimization of Pharmacokinetic Properties. ACS Med Chem Lett. 2022.

CAS Number: 1800343-11-6

Molecular Weight: 516.62

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Epigenetic Reader Domain
Mehr Informationen
Artikelnummer MEXHY-150516S-1
Hersteller MedChemExpress
Hersteller Artikelnummer HY-150516S-1
Verpackungseinheit 1 mg
Mengeneinheit STK
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