Darifenacin-d4, CAS 1095598-84-7

Product Description: Darifenacin-d4 is the deuterium labeled Darifenacin[1]. Darifenacin(UK88525) is a selective M3 muscarinic receptor antagonist with pKi of 8.9. IC50 value: 8.9 (pKi)[2].

Applications: Neuroscience-Neuromodulation

Formula: C28H26D4N2O2

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019 Feb;53(2):211-216./[2]Hegde SS, et al. Functional role of M2 and M3 muscarinic receptors in the urinary bladder of rats in vitro and in vivo. Br J Pharmacol, 1997, 120(8), 1409-1418.

CAS Number: 1095598-84-7

Molecular Weight: 430.57

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: mAChR

• Artikelnummer: MEXHY-A0033S1-1
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-A0033S1-1
• Verpackungseinheit: 1 mg
• Mengeneinheit: STK