Relebactam-d9

Product Description: Relebactam-d9 (MK-7655-d9) is deuterium labeled Relebactam. Relebactam is a diazabicyclooctane inhibitor with activity against a wide spectrum of β-lactamases, including class A (extended-spectrum β-lactamases and KPC) and class C (AmpC) enzymes. Relebactam shows antibacterial activity[1].

Applications: COVID-19-immunoregulation

Formula: C12H11D9N4O6S

References: [1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216./[2]Lapuebla A, et al. Activity of Imipenem with Relebactam against Gram-Negative Pathogens from New York City. Antimicrob Agents Chemother. 2015 Aug;59(8):5029-31./[3]Bush K. A resurgence of β-lactamase inhibitor combinations effective against multidrug-resistant Gram-negative pathogens. Int J Antimicrob Agents. 2015 Nov;46(5):483-93.

Molecular Weight: 357.43

Research Area: Infection

Target: Bacterial;Beta-lactamase;Isotope-Labeled Compounds

• Artikelnummer: MEXHY-16752S1-0
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-16752S1-0
• Verpackungseinheit: Get quote
• Mengeneinheit: STK