GSK-5959, CAS 901245-65-6

GSK-5959, CAS 901245-65-6
Artikelnummer
BPS82066
Verpackungseinheit
25 mg
Hersteller
BPS Bioscience

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CAS Number: 901245-65-6

Description: GSK-5959 exhibits >100-fold selectivity for BRPF1 (IC50 = 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression and have been implicated in human cancer.

Format: Solid

Storage Stability: At least 6 months at -20°C. 

Warnings: Avoid freeze/thaw cycles

Biosafety Level: Not applicable (BSL-1)
Mehr Informationen
Artikelnummer BPS82066
Hersteller BPS Bioscience
Hersteller Artikelnummer 82066
Green Labware Nein
Verpackungseinheit 25 mg
Mengeneinheit STK
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