NBI 98782, CAS 85081-18-1

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: (2R)-1,3R,4,6,7,11bR-hexahydro-9,10-dimethoxy-3-(2-methylpropyl)-2H-benzo[a]quinolizin-2-ol

Purity: ≥98%

Formula Markup: C19H29NO3

Formula Weight: 319.4385

CAS Number: 85081-18-1

Notes: An inhibitor of VMAT2 (Ki = 3.96 nM) and an active metabolite of tetrabenazine and valbenazine; selective for VMAT2 over a panel of 80 receptors at 10 µM; decreases dopamine, 5-HT, and norepinephrine levels and increases DOPAC, HVA, and 5-HIAA levels in the mouse medial prefrontal cortex at 10 mg/kg; induces ptosis and increases serum prolactin levels in rats at 10 mg/kg; inhibits PCP- and amphetamine-induced hyperactivity in mice at 10 mg/kg

• Artikelnummer: CAY42116-50
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 42116-50
• Verpackungseinheit: 50 mg
• Mengeneinheit: STK