BI-7273, CAS 1883429-21-7

Product Description: BI-7273 is a selective, and cell-permeable BRD9 inhibitor, with an IC50 and a Kd of 19 and 0.75 nM; also shows high effect on BRD7, with an IC50 and a Kd of 117 nM and 0.3 nM.

Applications: Cancer-Kinase/protease

Formula: C20H23N3O3

References: [1]Martin LJ, et al. Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor. J Med Chem. 2016 May 26;59(10):4462-75./[2]Laetitia J Martin, et al. Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor. J Med Chem. 2016 May 26;59(10):4462-75.

CAS Number: 1883429-21-7

Molecular Weight: 353.41

Compound Purity: 99.83

Research Area: Cancer

Solubility: DMSO : 10 mg/mL (ultrasonic)

Target: Epigenetic Reader Domain

• Artikelnummer: MEXHY-100351-100
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-100351-100
• Verpackungseinheit: 100 mg
• Mengeneinheit: STK