POI ligand 1

POI ligand 1
Artikelnummer
MEXHY-168864-0
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MedChemExpress

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Product Description: POI ligand 1 is a template for the non-selective HDAC inhibitor Vorinostat (HY-10221). POI ligand 1 can serve as a ligand for target protein (Ligands for Target Protein for PROTAC) for the development of PROTAC HDAC degraders with antitumor activity. POI ligand 1 can be used for the synthesis of FF2049 (HY-168863)[1].

Applications: Cancer-programmed cell death

Formula: C14H21N3O3

References: [1]Feller F, et al. Development of the First-in-Class FEM1B-Recruiting Histone Deacetylase Degraders. J Med Chem. 2025 Jan 13.

Molecular Weight: 279.33

Research Area: Cancer

Target: HDAC;Ligands for Target Protein for PROTAC
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Artikelnummer MEXHY-168864-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-168864-0
Verpackungseinheit Get quote
Mengeneinheit STK
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