PROTAC BRD4 Degrader-29

PROTAC BRD4 Degrader-29
Artikelnummer
MEXHY-172124-0
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MedChemExpress

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Product Description: PROTAC BRD4 Degrader-29 (compound 7a) is a potent PROTACs degrader of BRD4, with the DC50 of 89.4 nM. PROTAC BRD4 Degrader-29 plays an important role in cancer research (Pink: ligand for target protein (HY-13030); Black: linker (HY-172125); Blue: E3 ligase ligand (HY-103597))[1].

Formula: C58H61ClN10O9S2

References: [1]Andrew McGown, et al. Use of Aldehyde–Alkyne–Amine Couplings to Generate Medicinal Chemistry-Relevant Linkers. ACS Medicinal Chemistry Letters

Molecular Weight: 1141.75

Research Area: Cancer

Target: Epigenetic Reader Domain;PROTACs
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Artikelnummer MEXHY-172124-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-172124-0
Verpackungseinheit Get quote
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