QXG-6442

QXG-6442
Artikelnummer
MEXHY-170953-0
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MedChemExpress

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Product Description: QXG-6442 is a CK1α Molecular Glue Degrader. QXG-6442 exhibits CK1α degradation potency with a DC50 of 5.7 nM and a Dmax of 90%. QXG-6442 induces antiproliferative effects in MOLM-14 cell line[1].

Applications: Cancer-Kinase/protease

Formula: C21H17N5O4

References: [1]Geng Q, et al. Development of Potent and Selective CK1α Molecular Glue Degraders. J Med Chem. 2025 Feb 13;68(3):3180-3196.

Molecular Weight: 403.39

Research Area: Cancer

Target: Casein Kinase;Molecular Glues
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Artikelnummer MEXHY-170953-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-170953-0
Verpackungseinheit Get quote
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