RSK-IN-2, CAS 3011713-80-4

RSK-IN-2, CAS 3011713-80-4
Artikelnummer
MEXHY-173406-0
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MedChemExpress

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Product Description: RSK-IN-2 (Compound 3e) is a RSK inhibitor, with IC50 s of 37.89 nM (RSK2), 30.78 nM (RSK1), 20.51 nM (RSK3), 91.28 nM (RSK4). RSK-IN-2 inhibits tumor cell proliferation, induces apoptosis and causes cell cycle arrest in the G2/M phase[1].

Formula: C25H30ClN7O3

References: [1]Han C, et al. Discovery of 2,4-dianilinopyrimidine derivatives as novel p90 ribosomal S6 protein kinase (RSK) inhibitors. Eur J Med Chem. 2025 Jul 5;291:117590.

CAS Number: 3011713-80-4

Molecular Weight: 512.00

Research Area: Cancer

Target: Apoptosis;Ribosomal S6 Kinase (RSK)
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Artikelnummer MEXHY-173406-0
Hersteller MedChemExpress
Hersteller Artikelnummer HY-173406-0
Verpackungseinheit Get quote
Mengeneinheit STK
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