Giredestrant, CAS 1953133-47-5

Product Description: Giredestrant (GDC-9545), a non-steroidal estrogen receptor (ER) ligand, is an orally active and selective ER antagonist. Giredestrant potently competes with Estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity[1].

Applications: Cancer-programmed cell death

Formula: C27H31F5N4O

References: [1]C Metcalfe, et al. Abstract P5-04-07: GDC-9545: A novel ER antagonist and clinical candidate that combines desirable mechanistic and pre-clinical DMPK attributes

CAS Number: 1953133-47-5

Molecular Weight: 522.55

Compound Purity: 99.52

Research Area: Cancer

Solubility: DMSO : 50 mg/mL (ultrasonic)

Target: Estrogen Receptor/ERR

• Artikelnummer: MEXHY-109176-10.1
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-109176-10.1
• Verpackungseinheit: 10 mM/1 ml
• Mengeneinheit: STK