GRK5-IN-2, CAS 1642839-27-7

GRK5-IN-2, CAS 1642839-27-7
Artikelnummer
MEXHY-136561-10.1
Verpackungseinheit
10 mM/1 ml
Hersteller
MedChemExpress

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Product Description: GRK5-IN-2 (compound 707), a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor. GRK5-IN-2 regulates the expression and/or release of insulin and is useful for the metabolic disease research[1].

Applications: Metabolism-protein/nucleotide metabolism

Formula: C20H20N4O4

References: [1]Axel Ullrich (Prof. Dr.), et al. Imidazo[4,5-c]pyridine and pyrrolo[3,2-c]pyridine compounds as G-protein-coupled receptor kinase 5 (GRK5) modulators. EP2818472A1.

CAS Number: 1642839-27-7

Molecular Weight: 380.40

Compound Purity: 99.92

Research Area: Metabolic Disease

Solubility: DMSO : 62.5 mg/mL (ultrasonic;warming;heat to 60°C)

Target: G Protein-coupled Receptor Kinase (GRK)
Mehr Informationen
Artikelnummer MEXHY-136561-10.1
Hersteller MedChemExpress
Hersteller Artikelnummer HY-136561-10.1
Verpackungseinheit 10 mM/1 ml
Mengeneinheit STK
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