Product Description: GSK2256098 is a selective FAK kinase inhibitor, which inhibits growth and survival of pancreatic ductal adenocarcinoma cells.
Applications: Cancer-Kinase/protease
Formula: C20H23ClN6O2
References: [1]Zhang J, et al. A small molecule FAK kinase inhibitor, GSK2256098, inhibits growth and survival of pancreatic ductal adenocarcinoma cells. Cell Cycle. 2014;13(19):3143-9./[2]Thanapprapasr D, et al. PTEN Expression as a Predictor of Response to Focal Adhesion Kinase Inhibition in Uterine Cancer. Mol Cancer Ther. 2015 Jun;14(6):1466-75.
CAS Number: 1224887-10-8
Molecular Weight: 414.89
Compound Purity: 99.62
Research Area: Cancer
Solubility: DMSO : ≥ 30 mg/mL
Target: Apoptosis;FAK