HC-067047, CAS 883031-03-6

Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: 2-methyl-1-[3-(4-morpholinyl)propyl]-5-phenyl-N-[3-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide

Purity: ≥98%

Formula Markup: C26H28F3N3O2

Formula Weight: 471.5

CAS Number: 883031-03-6

Notes: HC-067047 is a TRPV4 antagonist that reversibly inhibits currents through human, rat, and mouse TRPV4 orthologs (IC50s = 48, 133, and 17 nM, respectively).{32658} It is selective for TRPV4 over TRPV1, TRPV2, TRPV3, and TRPM8 channels.{32658} HC-067047 has been shown to increase functional bladder capacity and to reduce micturition frequency in wild-type mice and rats with cystitis.{32658}

• Artikelnummer: CAY20927-5
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 20927-5
• Verpackungseinheit: 5 mg
• Mengeneinheit: STK