Description: MM 11253 is a RARγ antagonist with IC50 of 44nM.
CAS Number: 345952-44-5
Formula: C28H30O2S2
Molecular Weight: 462,67
References: M I Dawson, et al. Retinoic acid (RA) receptor transcriptional activation correlates with inhibition of 12-O-tetradecanoylphorbol-13-acetate-induced ornithine decarboxylase (ODC) activity by retinoids: a potential role for trans-RA-induced ZBP-89 in ODC inhibition. Int J Cancer. 2001 Jan 1;91(1):8-21.