Product Description: Orforglipron (LY3502970) (Compound 67) is an orally active agonist for Glucagon-like peptide-1 receptor (GLP-1R), which exhibits potency in ameliorates the type 2 diabete[1].
Applications: Metabolism-sugar/lipid metabolism
Formula: C48H48F2N10O5
References: [1]Pyrazolopyridine derivative having glp-1 receptor agonist effect. WO2018056453A1/[2]Kawai T, Sun B, Yoshino H, et al. Structural basis for GLP-1 receptor activation by LY3502970, an orally active nonpeptide agonist. Proc Natl Acad Sci U S A. 2020;117(47):29959-29967.
CAS Number: 2212020-52-3
Molecular Weight: 882.96
Compound Purity: 99.80
Research Area: Metabolic Disease
Solubility: DMSO : 50 mg/mL (ultrasonic;warming;heat to 60°C)
Target: GCGR