Product Description: P-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance.
Applications: Cancer-programmed cell death
Formula: C32H31N5O2
References: [1]Qiu Q, et al. Design, Synthesis, and Pharmacological Characterization of N-(4-(2 (6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)yl)ethyl)phenyl)quinazolin-4-amine Derivatives: Novel Inhibitors Reversing P-Glycoprotein-Mediated Multidrug Resistance. J Med Chem. 2017 Apr 27;60(8):3289-3302.
CAS Number: 2050747-49-2
Molecular Weight: 517.62
Compound Purity: 98.79
Research Area: Cancer
Solubility: DMSO : 16.67 mg/mL (ultrasonic;warming;heat to 70°C)
Target: P-glycoprotein