PD 81723, CAS 132861-87-1

PD 81723, CAS 132861-87-1
Artikelnummer
CAY42371-5
Verpackungseinheit
5 mg
Hersteller
Cayman Chemical

Verfügbarkeit: wird geladen...
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Shelf life (days): 1460.0

Formulation: A solid

Formal Name: (2-amino-4,5-dimethyl-3-thienyl)[3-(trifluoromethyl)phenyl]-methanone

Purity: ≥95%

Formula Markup: C14H12F3NOS

Formula Weight: 299.3

CAS Number: 132861-87-1

Notes: An adenosine A1 receptor positive allosteric modulator; inhibits TNF-a and cycloheximide-induced apoptosis in HK-2 kidney epithelial cells at 10 µM; increases right atrial heart rate in combination with ADA in isolated rat right atria (EC50 = 0.83 nM); reduces plasma creatinine levels and infarct area in a mouse model of renal ischemia-reperfusion injury at 3 mg/kg
Mehr Informationen
Artikelnummer CAY42371-5
Hersteller Cayman Chemical
Hersteller Artikelnummer 42371-5
Verpackungseinheit 5 mg
Mengeneinheit STK
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