PF-750, CAS 959151-50-9

PF-750, CAS 959151-50-9
Artikelnummer
CAY10010908-5
Verpackungseinheit
5 mg
Hersteller
Cayman Chemical

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Shelf life (days): 1460.0

Formulation: A crystalline solid

Formal Name: N-phenyl-4-(quinolin-2-ylmethyl)piperidine-1-carboxamide

Purity: ≥98%

Formula Markup: C22H23N3O

Formula Weight: 345.4

CAS Number: 959151-50-9

Notes: Fatty acid amide hydrolase (FAAH) is the enzyme responsible for hydrolysis and inactivation of fatty acid amides including anandamide and oleamide. PF-750 is a potent, time-dependent, irreversible FAAH inhibitor with IC50 values of 0.6 and 0.016 µM when preincubated with recombinant human FAAH for 5 and 60 minutes, respectively.{15092} Activity-based profiling of various human and murine tissue proteome samples revealed that PF-750 is highly selective for FAAH relative to other serine hydrolases, showing no discernable off-site activity up to 500 µM.{15092}
Mehr Informationen
Artikelnummer CAY10010908-5
Hersteller Cayman Chemical
Hersteller Artikelnummer 10010908-5
Verpackungseinheit 5 mg
Mengeneinheit STK
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