Product Description: PKA-IN-1 is a potent and selective cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor with an IC50 of 0.03 μM[1].
Applications: COVID-19-immunoregulation
Formula: C13H11N3O
References: [1]Z X Lu, et al. Selective inhibition of cyclic AMP-dependent protein kinase by isoquinoline derivative. Biol Chem Hoppe Seyler. 1996 Jun;377(6):373-8
CAS Number: 179985-52-5
Molecular Weight: 225.25
Compound Purity: 99.88
Research Area: Inflammation/Immunology
Solubility: DMSO : 62.5 mg/mL (ultrasonic;warming;heat to 80°C)