Revefenacin, CAS 864750-70-9

Product Description: Revefenacin (TD-4208; GSK1160724) is a potent mAChR antagonist; has a high affinity on M3 receptor with a Ki of 0.18 nM.

Applications: COVID-19-immunoregulation

Formula: C35H43N5O4

References: [1]Steinfeld T, et al. In vitro characterization of TD-4208, a lung-selective and long-acting muscarinic antagonist bronchodilator (Abstract). Am J Respir Crit Care Med 179:A4553./[2]Pulido-Rios MT, et al. In vivo pharmacological characterization of TD-4208, a novel lung-selective inhaled muscarinic antagonist with sustained bronchoprotective effect in experimental animal models. J Pharmacol Exp Ther. 2013 Aug;346(2):241-50.

CAS Number: 864750-70-9

Molecular Weight: 597.75

Compound Purity: 99.23

Research Area: Inflammation/Immunology; Cardiovascular Disease

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: mAChR

• Artikelnummer: MEXHY-15851-10.1
• Hersteller: MedChemExpress
• Hersteller Artikelnummer: HY-15851-10.1
• Verpackungseinheit: 10 mM/1 ml
• Mengeneinheit: STK