T-3775440 hydrochloride, CAS 1422535-52-1

T-3775440 hydrochloride, CAS 1422535-52-1
Artikelnummer
MEXHY-103085-10.1
Verpackungseinheit
10 mM/1 ml
Hersteller
MedChemExpress

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Product Description: T-3775440 (hydrochloride) is an irreversible lysine-specific histone demethylase (LSD1) inhibitor with an IC50 value of 2.1 nM.

Applications: Cancer-programmed cell death

Formula: C18H23ClN4O

References: [1]Ishikawa Y, et al. A Novel LSD1 Inhibitor T-3775440 Disrupts GFI1B-Containing Complex Leading to Transdifferentiation and Impaired Growth of AML Cells. Mol Cancer Ther. 2017 Feb;16(2):273-284.

CAS Number: 1422535-52-1

Molecular Weight: 346.85

Compound Purity: 99.13

Research Area: Cancer

Solubility: DMSO : ≥ 30.18 mg/mL/H2O : 8.33 mg/mL (ultrasonic;warming;heat to 60°C)

Target: Histone Demethylase
Mehr Informationen
Artikelnummer MEXHY-103085-10.1
Hersteller MedChemExpress
Hersteller Artikelnummer HY-103085-10.1
Verpackungseinheit 10 mM/1 ml
Mengeneinheit STK
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