Taspoglutide (acetate), CAS 1022150-16-8

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: 8-(2-methylalanine)-35-(2-methylalanine)-36-L-argininamide-7-36-glucagon-like peptide I (human), acetate

Amino Acids: HXEGTFTSDVSSYLEGQAAKEFIAWLVKXR-NH2 (X = α-aminoiso

Purity: ≥98%

Formula Markup: C152H232N40O45 / XC2H4O2

Formula Weight: 3339.71108

CAS Number: 1022150-16-8

Notes: Taspoglutide is an agonist of the glucagon-like peptide 1 receptor (GLP-1R; Ki = 1.1 nM for the human receptor).{67869} It induces cAMP accumulation in CHO-K1 cells expressing human GLP-1R (EC50 = 0.06 nM). Taspoglutide (1 mg/animal per week) decreases blood levels of glucose and increases blood levels of insulin in an oral glucose tolerance test in Zucker diabetic obese rats. It reduces blood levels of gastric inhibitory polypeptide (GIP), plasma levels of triglycerides, and body weight in the same model.{67870}

• Artikelnummer: CAY41258-10
• Hersteller: Cayman Chemical
• Hersteller Artikelnummer: 41258-10
• Verpackungseinheit: 10 mg
• Mengeneinheit: STK