Product Description: TG 100713 is an inhibitor of PI3K, with IC50s of 24, 50, 165, and 215 nM for PI3Kδ, γ, α and β isoforms respectively[1].
Applications: Cancer-Kinase/protease
Formula: C12H10N6O
References: [1]Doukas J, et, al. Phosphoinositide 3-kinase gamma/delta inhibition limits infarct size after myocardial ischemia/reperfusion injury. Proc Natl Acad Sci U S A. 2006 Dec 26;103(52):19866-71.
CAS Number: 925705-73-3
Molecular Weight: 254.25
Compound Purity: 99.49
Research Area: Cancer
Solubility: DMSO : 6.41 mg/mL (ultrasonic)
Target: PI3K