VT103, CAS 2290608-13-6

VT103, CAS 2290608-13-6
Artikelnummer
CAY42327-10
Verpackungseinheit
10 mg
Hersteller
Cayman Chemical

Verfügbarkeit: wird geladen...
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Shelf life (days): 1460.0

Formulation: A solid

Formal Name: N-methyl-3-(1-methyl-1H-imidazol-4-yl)-4-[[4-(trifluoromethyl)phenyl]amino]-benzenesulfonamide

Purity: ≥98%

Formula Markup: C18H17F3N4O2S

Formula Weight: 410.414549

CAS Number: 2290608-13-6

Notes: A TEAD1 inhibitor (IC50 = 1.02 nM); inhibits TEAD autopalmitoylation in HEK293 cells expressing TEAD1 but not HEK293 cells expressing TEAD2, TEAD3, or TEAD4 at 3 µM; inhibits palmitoylation of endogenous TEAD1 in NCI-H2373 cells; reduces tumor volume in NCI-H2373 and NCI H226 mesothelioma mouse xenograft models
Mehr Informationen
Artikelnummer CAY42327-10
Hersteller Cayman Chemical
Hersteller Artikelnummer 42327-10
Verpackungseinheit 10 mg
Mengeneinheit STK
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