MU1210, CAS 2275601-87-9

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: 5-(1-methyl-1H-pyrazol-4-yl)-3-[3-(4-pyridinyl)phenyl]-furo[3,2-b]pyridine

Purity: ≥95%

Formula Markup: C22H16N4O

Formula Weight: 352.4

CAS Number: 2275601-87-9

Notes: MU1210 is an inhibitor of CDC-like kinase 1 (Clk1), Clk2, and Clk4 (IC50s = 8, 20, and 12 nM, respectively).{72474} It is selective for these kinases over Clk3 (IC50 = >3,000 nM), as well as dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A), DYRK1B, DYRK2, homeodomain-interacting protein kinase 1 (HIPK1), and HIPK3 (IC50s = 213, 956, 1,309, 187, and 159 nM, respectively) but does inhibit HIPK2 (IC50 = 23 nM).

• SKU: CAY41308-1
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 41308-1
• Package Unit: 1 mg
• Quantity Unit: STK