AG-045572, CAS 263847-55-8

Shelf life (days): 1460.0

Formulation: A solid

Formal Name: 5-[(5,6,7,8-tetrahydro-3,5,5,8,8-pentamethyl-2-naphthalenyl)methyl]-N-(2,4,6-trimethoxyphenyl)-2-furancarboxamide

Purity: ≥98%

Formula Markup: C30H37NO5

Formula Weight: 491.6

CAS Number: 263847-55-8

Notes: A GnRH receptor antagonist (Kis = 6, 2.2, and 3.8 nM for the human, mouse, and rat receptors, respectively); selective for the GnRH receptor over a panel of 43 receptors, ion channels, and enzymes at 1 µM; prevents GnRH-induced increases in inositol phosphate production in HEK293 cells expressing the human GnRH receptor (KB = 25 nM); oral or intravenous administration decreases plasma LH levels in castrated rats; inhibits GnRH-A-induced increases in plasma LH and testosterone levels in non-castrated rats at 20 mg/kg

• SKU: CAY42244-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 42244-10
• Package Unit: 10 mg
• Quantity Unit: STK