ALK inhibitor 1, CAS 761436-81-1

ALK inhibitor 1, CAS 761436-81-1
SKU
MEXHY-15357-10.1
Packaging Unit
10 mM/1 ml
Manufacturer
MedChemExpress

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Product Description: ALK inhibitor 1 (compound 17) is a potent pyrimidin ALK inhibitor. ALK inhibitor 1 is a potent inhibitor of testis-specific serine/threonine kinase 2 (TSSK2; IC50=31 nM) and focal adhesion kinase (FAK; IC50=2 nM)[1].

Applications: Cancer-Kinase/protease

Formula: C23H28BrN7O3S

References: [1]Jon E Hawkinson, et al. Potent Pyrimidine and Pyrrolopyrimidine Inhibitors of Testis-Specific Serine/Threonine Kinase 2 (TSSK2). ChemMedChem. 2017 Nov 22;12(22):1857-1865.

CAS Number: 761436-81-1

Molecular Weight: 562.48

Compound Purity: 99.62

Research Area: Cancer

Solubility: 1M HCl : 100 mg/mL (ultrasonic;adjust pH to 1 with HCl)/DMSO : ≥ 100 mg/mL

Target: Anaplastic lymphoma kinase (ALK);FAK
More Information
SKU MEXHY-15357-10.1
Manufacturer MedChemExpress
Manufacturer SKU HY-15357-10.1
Package Unit 10 mM/1 ml
Quantity Unit STK
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