Product Description: Apinocaltamide (ACT-709478) is a potent, selective, orally active, and brain penetrating T-type calcium channel blocker. ACT-709478 is used in the research of generalized epilepsies[1].
Applications: Neuroscience-Neuromodulation
Formula: C22H18F3N5O
References: [1]Bezençon O, et al. Discovery of a Potent, Selective T-type Calcium Channel Blocker as a Drug Candidate for the Treatment of Generalized Epilepsies. J Med Chem. 2017 Dec 14;60(23):9769-9789.
CAS Number: 1838651-58-3
Molecular Weight: 425.41
Compound Purity: 99.83
Research Area: Neurological Disease
Solubility: DMSO : ≥ 125 mg/mL
Target: Calcium Channel