Product Description: ASP-9521 is a potent, selective and orally available AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.
Applications: Cancer-programmed cell death
Formula: C19H26N2O3
References: [1]Kikuchi A, et al. In vitro and in vivo characterisation of ASP9521: a novel, selective, orally bioavailable inhibitor of 17β-hydroxysteroid dehydrogenase type 5 (17βHSD5; AKR1C3).Invest New Drugs. 2014 Oct;32(5):860-70.
CAS Number: 1126084-37-4
Molecular Weight: 330.42
Compound Purity: 98.0
Research Area: Cancer
Solubility: DMSO : 100 mg/mL (ultrasonic)
Target: Others