BIM5078, CAS 337506-43-1

Product Description: BIM5078 is a hepatocyte nuclear factor 4α (HNF4α) antagonist that can inhibit the expression of known HNF4α target genes. BIM5078 represses insulin promoter activity through HNF4α antagonism. BIM5078 can be used for the research of cancer and diabetes[1].

Applications: Metabolism-protein/nucleotide metabolism

Formula: C14H10ClN3O4S

References: [1]Kiselyuk A, et al. HNF4α antagonists discovered by a high-throughput screen for modulators of the human insulin promoter. Chem Biol. 2012 Jul 27;19(7):806-18.

CAS Number: 337506-43-1

Molecular Weight: 351.76

Research Area: Cancer; Metabolic Disease

Solubility: 10 mM in DMSO

Target: Nuclear Hormone Receptor 4A/NR4A

• SKU: MEXHY-119971-25
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-119971-25
• Package Unit: 25 mg
• Quantity Unit: STK