BRD9539, CAS 1374601-41-8

Product Description: BRD9539 is a histone methyltransferase G9a inhibitor with an IC50 of 6.3 μM. BRD9539 also inhibits PRC2 activity and is inactive against SUV39H1, NSD2 and DNMT1[1].

Applications: Cancer-Kinase/protease

Formula: C24H21N3O3

References: [1]Yuan Y et al. A small-molecule probe of the histone methyltransferase G9a induces cellular senescence in pancreatic adenocarcinoma. ACS Chem Biol. 2012 Jul 20;7(7):1152-7.

CAS Number: 1374601-41-8

Molecular Weight: 399.44

Compound Purity: 99.74

Research Area: Cancer

Solubility: DMSO : 16.67 mg/mL (ultrasonic)

Target: Histone Methyltransferase

• SKU: MEXHY-15647-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-15647-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK