Product Description: CB1 inverse agonist 2 is an orally active inverse agonist of Cannabinoid Receptor CB1. CB1 inverse agonist 2 effectively inhibits CP55940-induced hypothermia and anorexia in mice model[1].
Applications: Neuroscience-Neuromodulation
Formula: C24H20ClFN2OS
References: [1]Synthesis and Evaluation of Dibenzothiazepines: A Novel Class of Selective Cannabinoid-1 Receptor Inverse Agonists
J. Med. Chem., 2009, 52 (7), pp 1975-1982/[2]Pettersson H, et al. Synthesis and evaluation of dibenzothiazepines: a novel class of selective cannabinoid-1 receptor inverse agonists. J Med Chem. 2009 Apr 9;52(7):1975-82.
CAS Number: 1019839-52-1
Molecular Weight: 438.94
Research Area: Neurological Disease
Solubility: 10 mM in DMSO
Target: Cannabinoid Receptor