CCG215022, CAS 1813527-81-9

Product Description: CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, GRK5 and GRK1, respectively.

Applications: Cancer-Kinase/protease

Formula: C26H22FN7O3

References: [1]Homan KT, et al. Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally DesignedInhibitor. J Biol Chem. 2015 Aug 21;290(34):20649-59.

CAS Number: 1813527-81-9

Molecular Weight: 499.50

Compound Purity: 98.69

Research Area: Cancer

Solubility: DMSO : ≥ 28 mg/mL

Target: PKA

• SKU: MEXHY-18991-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-18991-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK