Conteltinib (tetrahydrochloride)

Conteltinib (tetrahydrochloride)
SKU
MEXHY-109084A-50
Packaging Unit
50 mg
Manufacturer
MedChemExpress

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Product Description: Conteltinib tetrahydrochloride (CT-707 tetrahydrochloride) is the tetrahydrochloride salt form of Conteltinib (HY-109084). Conteltinib tetrahydrochloride is the inhibitor for FAK (IC50=1.6 nM), ALK, and Pyk2. Conteltinib tetrahydrochloride exhibits a synergistic anti-tumor efficacy with Cabozantinib (HY-13016)[1].

Formula: C32H49Cl4N9O3S

References: [1]Wang DD, et al. CT-707, a Novel FAK Inhibitor, Synergizes with XL184 to Suppress Hepatocellular Carcinoma by Blocking XL184-Induced FAK Activation. Mol Cancer Ther. 2016 Dec;15(12):2916-2925.

Molecular Weight: 781.67

Compound Purity: 99.60

Research Area: Cancer

Target: FAK
More Information
SKU MEXHY-109084A-50
Manufacturer MedChemExpress
Manufacturer SKU HY-109084A-50
Package Unit 50 mg
Quantity Unit STK
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