Shelf life (days): 1095.0
Formulation: A neat solid
Formal Name: 3-(5H-dibenzo[a,d]cyclohepten-5-ylidene)-N,N-dimethyl-1-propanamine, monohydrochloride
Purity: ≥98%
Formula Markup: C20H21N / HCl
Formula Weight: 311.9
CAS Number: 6202-23-9
Notes: Cyclobenzaprine is a skeletal muscle relaxant that also has sedative properties.{25863,25864,25861} It has been shown to antagonize muscarinic receptors (Kis = 25, 60, and 6 nM for M1, M2, and M3, respectively), serotonin 5-HT2 receptors (Kis = 56 and 330 nM for 5-HT2C and 5-HT2B, respectively), and histamine H1 receptor (IC50 = 20 nM).{25917,25919,25918}