Enerisant, CAS 1152747-82-4

Product Description: Enerisant (TS-091) is a potent, highly selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2.89 nM and 14.5 nM against human and rat histamine H3 receptors, respectively[1].

Applications: Neuroscience-Neuromodulation

Formula: C22H30N4O3

References: [1]Hino N, et al. A novel potent and selective histamine H3 receptor antagonist enerisant: in vitro profiles, in vivo receptor occupancy, and wake-promoting and procognitive effects in rodents. Journal of Pharmacology and Experimental Therapeutics, 2020, 375(2): 276-285.

CAS Number: 1152747-82-4

Molecular Weight: 398.50

Compound Purity: 99.79

Research Area: Neurological Disease

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: Histamine Receptor

• SKU: MEXHY-17610-10.1
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-17610-10.1
• Package Unit: 10 mM/1 ml
• Quantity Unit: STK